SCHEMBL16339443

SCHEMBL16339443

Cn1ccc2cc(-c3cnc(N)nc3N)ccc21

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.56
LRRK2 Q5S007 2/20 0.54
PIK3CB P42338 2/20 0.49
PRKCI P41743 1/20 0.49
SRC P12931 5/20 0.46
ABL1 P00519 3/20 0.46
PIK3CD O00329 1/20 0.46
EGFR P00533 1/20 0.46
HCK P08631 1/20 0.46
KDR P35968 1/20 0.46
PIK3CA P42336 1/20 0.46
MTOR P42345 1/20 0.46
PIK3CG P48736 1/20 0.46
EPHB4 P54760 1/20 0.46
PRKDC P78527 1/20 0.46
HSD11B1 P28845 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12612181 0.89 DHFR (0.56) DHFRLRRK2PIK3CB
SCHEMBL10181112 0.78 DHFR (0.50) DHFRSRCKDR
SCHEMBL4474184 0.75 DHFR (0.50) DHFRKDR
SCHEMBL3838310 0.74 DHFR (0.56) DHFR
SCHEMBL29430406 0.74 DHFR (0.52) DHFRKDR
SCHEMBL4463726 0.74 DHFR (0.52) DHFRKDR
Hydrochloric Acid SCHEMBL4473311 0.73 DHFR (0.55) DHFRSRC
SCHEMBL3564713 0.72 BTK (0.49) LRRK2PRKCISRCABL1EGFR
SCHEMBL28342224 0.72 DHFR (1.00) DHFRKDR
SCHEMBL30556294 0.72 DHFR (1.00) DHFRKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8927547-B2 Pyrimidine derivatives NOVIGA RESEARCH AB (SE) 2015-01-06 US claimed
EP-2688883-B1 PYRIMIDINE DERIVATIVES NOVIGA RES AB (SE) 2016-05-18 EP disclosed