SCHEMBL16346231

SCHEMBL16346231

COc1ccc(C=O)cc1-c1cc2c(NCCc3ccccc3)ncnc2s1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.71
MAPK1 P28482 1/20 0.52
NPC1 O15118 1/20 0.52
GALR3 O60755 1/20 0.52
NR2F2 P24468 1/20 0.52
RAB9A P51151 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16375358 0.83 EGFR (1.00) EGFR
SCHEMBL16345771 0.81 EGFR (0.70) EGFR
SCHEMBL16346230 0.81 EGFR (1.00) EGFR
SCHEMBL16376056 0.76 EGFR (1.00) EGFRMAPK1
SCHEMBL5435953 0.76 EGFR (0.53) EGFRMAPK1NPC1RAB9A
SCHEMBL16346492 0.75 EGFR (0.70) EGFR
SCHEMBL16376005 0.73 EGFR (0.86) EGFR
SCHEMBL16345769 0.73 EGFR (0.77) EGFR
SCHEMBL5431882 0.72 ICAM1 (0.59) EGFRMAPK1NPC1GALR3NR2F2
SCHEMBL5433413 0.70 ICAM1 (0.77) EGFRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015000959-A1 4-AMINO-6-ARYL[2,3-D]PYRIMIDINES FOR THE INHIBITION OF EGFR TYROSINE KINASE NORWEGIAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (NTNU) (NO) 2015-01-08 WO disclosed