SCHEMBL16375358

SCHEMBL16375358

COc1cc(C=O)ccc1-c1cc2c(NCc3ccccc3)ncnc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 1.00
ICAM1 P05362 1/20 0.52
SELE P16581 1/20 0.52
VCAM1 P19320 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16376056 0.85 EGFR (1.00) EGFR
SCHEMBL16376062 0.85 EGFR (1.00) EGFRICAM1SELEVCAM1
SCHEMBL16346231 0.83 EGFR (0.71) EGFR
SCHEMBL16345771 0.82 EGFR (0.70) EGFR
SCHEMBL16376005 0.82 EGFR (0.86) EGFR
SCHEMBL16345769 0.81 EGFR (0.77) EGFR
SCHEMBL16376022 0.80 EGFR (0.67) EGFR
SCHEMBL16345767 0.78 EGFR (0.67) EGFR
SCHEMBL16346230 0.75 EGFR (1.00) EGFR
SCHEMBL16375362 0.74 EGFR (0.82) EGFRICAM1SELEVCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015000959-A1 4-AMINO-6-ARYL[2,3-D]PYRIMIDINES FOR THE INHIBITION OF EGFR TYROSINE KINASE NORWEGIAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (NTNU) (NO) 2015-01-08 WO disclosed