SCHEMBL1635209

SCHEMBL1635209

C=CCCCC(=O)NCCN1Cc2cc(Br)ccc2N=C1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.38
BACE2 Q9Y5Z0 1/20 0.34
TSHR P16473 1/20 0.33
HDAC6 Q9UBN7 3/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
PDE4A P27815 10/20 0.33
PDE4B Q07343 10/20 0.33
PDE4C Q08493 10/20 0.33
PDE4D Q08499 10/20 0.33
NPC1 O15118 1/20 0.32
NAMPT P43490 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1634599 0.86 BACE1 (0.39) BACE1BACE2TSHRHDAC3HDAC1
SCHEMBL8266027 0.85 BACE1 (0.41) BACE1BACE2TSHRPDE4APDE4B
SCHEMBL1635144 0.82 BACE1 (0.38) BACE1BACE2HDAC6HDAC3HDAC4
SCHEMBL8265789 0.78 DRD2 (0.43) BACE1BACE2PDE4APDE4BPDE4C
SCHEMBL13176987 0.77 BACE1 (0.35) BACE1BACE2PDE4APDE4BPDE4C
SCHEMBL8265973 0.75 BACE1 (0.44) BACE1TSHRPDE4APDE4BPDE4C
SCHEMBL1634699 0.75 BACE2 (0.43) BACE1BACE2PDE4APDE4BPDE4C
SCHEMBL13114389 0.73 BACE1 (0.40) BACE1PDE4APDE4BPDE4CPDE4D
SCHEMBL5350869 0.71 PDE4A (0.48) BACE1BACE2PDE4APDE4BPDE4C
SCHEMBL14723904 0.70 BACE1 (0.50) BACE1HDAC6HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7932261-B2 Macrocycle derivatives useful as inhibitors of β-secretase (BACE) JANSSEN PHARMACEUTICA NV (BE) 2011-04-26 US disclosed