SCHEMBL16355449

SCHEMBL16355449

CN[C@H](C)c1ncc(-c2ccc(Br)cc2)[nH]1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.43
TRPV1 Q8NER1 1/20 0.42
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
EGFR P00533 3/20 0.39
HDAC1 Q13547 1/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16355444 1.00 PTGES (0.43) PTGESTRPV1CCNB2CDK1CCNB1
SCHEMBL12158461 0.90 NPC1 (0.37)
SCHEMBL16355447 0.86 CDK5 (0.41) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL16355442 0.84 SCN10A (0.36)
SCHEMBL19323265 0.81 TRPV1 (0.44) PTGESTRPV1EGFR
SCHEMBL14300085 0.81 NPC1 (0.34) HDAC1
SCHEMBL12107457 0.81 NLN (0.41) GSK3BHDAC1
SCHEMBL14274103 0.81 SCN5A (0.34)
SCHEMBL16355456 0.80 CYP1A1 (0.37) HDAC1
SCHEMBL14708714 0.79 HDAC1 (0.43) PTGESTRPV1CCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140378416-A1 SILYL-CONTAINING HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME CORP. 2014-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140378416-A1 SILYL-CONTAINING HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES ZC3HAV1L, HBS1L, HAVCR2 PTGES 2608/4885TRPV1 4314/4885CCNB2 472/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.