SCHEMBL16358403

SCHEMBL16358403

C=C(OCC)c1cccc(CN2CCN(C)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.49
HDAC3 O15379 3/20 0.47
HDAC4 P56524 3/20 0.47
HDAC1 Q13547 3/20 0.47
HDAC7 Q8WUI4 3/20 0.47
HDAC2 Q92769 3/20 0.47
HDAC10 Q969S8 3/20 0.47
HDAC11 Q96DB2 3/20 0.47
HDAC8 Q9BY41 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
HDAC9 Q9UKV0 3/20 0.47
HDAC5 Q9UQL6 3/20 0.47
KDM4E B2RXH2 3/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CHRM3 P20309 1/20 0.46
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
HIF1A Q16665 1/20 0.44
ALDH1A1 P00352 2/20 0.43
FAAH O00519 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14387318 0.84 PRMT1 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24799638 0.82 MC4R (0.53) MC4RHDAC3HDAC4HDAC1HDAC7
SCHEMBL3453981 0.76 CYP2D6 (0.73) MC4RHDAC3HDAC4HDAC1HDAC7
SCHEMBL1481516 0.76 HDAC6 (0.58) MC4RHDAC3HDAC4HDAC1HDAC7
SCHEMBL31721203 0.76 CYP2D6 (0.73) MC4RHDAC3HDAC4HDAC1HDAC7
SCHEMBL13535291 0.76 MC4R (0.74) MC4RKDM4EALDH1A1MAPTCHKA
SCHEMBL10145077 0.76 ALDH1A1 (0.60) MC4RHDAC3HDAC4HDAC1HDAC7
SCHEMBL31721209 0.76 ALDH1A1 (0.60) MC4RHDAC3HDAC4HDAC1HDAC7
SCHEMBL16358261 0.75 HDAC6 (0.52) MC4RHDAC3HDAC4HDAC1HDAC7
SCHEMBL608151 0.75 CYP2D6 (0.54) HDAC1KDM4ECYP2D6CYP2C9HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007137196-A2 TUBULIN BINDING ANTI CANCER COMPOUNDS AND PRODRUGS THEREOF THRESHOLD PHARMACEUTICALS, INC. (US) 2007-11-29 WO disclosed