SCHEMBL1635888

SCHEMBL1635888

c1ccc(COc2cccc(CCNC3CCCCC3)c2)cc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FOXM1 Q08050 1/20 0.58
TAAR1 Q96RJ0 1/20 0.57
KDM4E B2RXH2 2/20 0.56
KMT2A Q03164 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
BCHE P06276 7/20 0.56
CYP4F2 P78329 1/20 0.54
CYP4A11 Q02928 1/20 0.54
CYP2D6 P10635 1/20 0.49
KDM1A O60341 1/20 0.49
ALDH1A1 P00352 2/20 0.49
SPHK2 Q9NRA0 1/20 0.47
SPHK1 Q9NYA1 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL69474 0.83 BCHE (0.51) FOXM1BCHECYP4F2CYP4A11CYP2D6
SCHEMBL12204184 0.82 ALDH1A1 (0.72) TAAR1KDM4EALDH1A1
SCHEMBL787022 0.81 ALDH1A1 (0.74) TAAR1KDM4EALDH1A1
SCHEMBL3665298 0.80 TAAR1 (0.84) TAAR1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL22216853 0.80 TAAR1 (0.84) TAAR1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL25002632 0.80 TAAR1 (0.84) TAAR1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL21792273 0.80 TAAR1 (0.84) TAAR1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL24767088 0.80 TAAR1 (0.84) TAAR1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL24075499 0.80 TAAR1 (0.84) TAAR1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL1240954 0.80 TAAR1 (0.84) TAAR1KMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7932261-B2 Macrocycle derivatives useful as inhibitors of β-secretase (BACE) JANSSEN PHARMACEUTICA NV (BE) 2011-04-26 US disclosed
US-20070232630-A1 MACROCYCLE DERIVATIVES USEFUL AS INHIBITORS OF beta-SECRETASE (BACE) JANSSEN PHARMACEUTICA NV (BE) 2007-10-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232630-A1 MACROCYCLE DERIVATIVES USEFUL AS INHIBITORS OF beta-SECRETASE (BACE) BACE2, BACE1, PSEN2 FOXM1 4180/4885TAAR1 4711/4885KDM4E 3557/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.