SCHEMBL1636732

SCHEMBL1636732

CN1C(=O)N(c2cccnc2F)C[C@H]1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 19/20 0.45
SCN9A Q15858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1636796 1.00 P2RX7 (0.45) P2RX7SCN9A
SCHEMBL1637705 0.89 P2RX7 (0.53) P2RX7
SCHEMBL1637645 0.87 P2RX7 (0.56) P2RX7
SCHEMBL1636775 0.83 P2RX7 (0.49) P2RX7
SCHEMBL2841345 0.83 P2RX7 (0.49) P2RX7
SCHEMBL1636701 0.82 P2RX7 (0.47) P2RX7
SCHEMBL1637472 0.81 P2RX7 (0.53) P2RX7
SCHEMBL1636761 0.81 P2RX7 (0.51) P2RX7
SCHEMBL1635930 0.77 P2RX7 (0.50) P2RX7
SCHEMBL1636103 0.76 P2RX7 (0.53) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7932282-B2 Imidazolidine carboxamide derivatives as P2X7 modulators GLAXO GROUP LIMITED (GB) 2011-04-26 US disclosed
CN-101679291-A Imidazolidine carboxamide derivatives as P2X7 modulators GLAXO GROUP LTD 2010-03-24 CN disclosed