SCHEMBL16369486

SCHEMBL16369486

CC(=O)c1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4cncnc4)CC3)cc2)c(CF)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 5/20 0.51
PTGER4 P35408 2/20 0.37
PTGER2 P43116 1/20 0.37
CNR1 P21554 1/20 0.36
MAPK14 Q16539 4/20 0.36
F10 P00742 1/20 0.35
CYP3A4 P08684 2/20 0.34
MMP13 P45452 2/20 0.34
MMP2 P08253 1/20 0.34
STAT3 P40763 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GSK3B P49841 2/20 0.34
CXCR4 P61073 1/20 0.34
KDM1A O60341 1/20 0.34
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16368731 0.89 BDKRB1 (0.49) BDKRB1PTGER4PTGER2CNR1MAPK14
SCHEMBL765546 0.89 BDKRB1 (0.53) BDKRB1PTGER4PTGER2CNR1MAPK14
SCHEMBL16369343 0.87 BDKRB1 (0.49) BDKRB1PTGER4PTGER2CNR1MAPK14
SCHEMBL765146 0.87 BDKRB1 (0.50) BDKRB1PTGER4PTGER2CNR1MAPK14
SCHEMBL12239063 0.86 BDKRB1 (0.60) BDKRB1CNR1MAPK14F10CYP3A4
SCHEMBL12239081 0.86 BDKRB1 (0.52) BDKRB1PTGER4PTGER2CNR1MAPK14
SCHEMBL10121331 0.82 BDKRB1 (0.60) BDKRB1CNR1MAPK14CYP3A4MMP13
SCHEMBL10121385 0.81 BDKRB1 (0.53) BDKRB1PTGER4PTGER2CNR1MAPK14
SCHEMBL12239059 0.81 BDKRB1 (0.53) BDKRB1PTGER4PTGER2CNR1MAPK14
SCHEMBL12262806 0.81 BDKRB1 (0.55) BDKRB1PTGER4PTGER2CNR1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8916589-B2 Bradykinin B1-antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-12-23 US disclosed