SCHEMBL16375008

SCHEMBL16375008

CCCCOc1c(C=O)ncc(C(=O)NCc2ccc(F)cc2F)c1ON

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.44
KCNA5 P22460 2/20 0.41
KCNK3 O14649 1/20 0.41
KCNK5 O95279 1/20 0.41
KCNK17 Q96T54 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41
PPARD Q03181 5/20 0.40
PDE10A Q9Y233 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PPARA Q07869 3/20 0.39
FAAH O00519 1/20 0.38
GSK3B P49841 1/20 0.38
CNR2 P34972 2/20 0.38
CCNE2 O96020 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
P2RX7 Q99572 2/20 0.37
JAK3 P52333 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15978569 0.89 MET (0.43) METKCNA5KCNK3KCNK5KCNK17
SCHEMBL16375007 0.77 MET (0.46) METKCNA5KCNK3KCNK5KCNK17
SCHEMBL16374956 0.77 PPARD (0.46) METKCNA5KCNK3KCNK5KCNK17
SCHEMBL8981574 0.76 CNR2 (0.52) FAAHCNR2
SCHEMBL16374958 0.76 KCNK3 (0.44) METKCNA5KCNK3KCNK5KCNK17
SCHEMBL15015195 0.75 PDE10A (0.42) METKCNA5KCNK3KCNK5KCNK17
SCHEMBL92991 0.75 CNR2 (0.49) FAAHCNR2
SCHEMBL19625793 0.73 KCNA5 (0.52) METKCNA5KCNK3KCNK5KCNK17
SCHEMBL2601314 0.71 PDE10A (0.49) METKCNA5KCNK3KCNK5KCNK17
SCHEMBL15015194 0.70 PDE10A (0.43) METKCNA5KCNK3KCNK5KCNK17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015001572-A2 PROCESS FOR THE PREPARATION OF INTERMEDIATE OF DOLUTEGRAVIR HETERO RESEARCH FOUNDATION (IN) 2015-01-08 WO disclosed