SCHEMBL16380712

SCHEMBL16380712

NC(=O)c1ccc(CO)c(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.47
EPHX2 P34913 2/20 0.40
HDAC6 Q9UBN7 1/20 0.40
VNN1 O95497 1/20 0.40
ERN1 O75460 1/20 0.40
PARP1 P09874 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
PDK2 Q15119 2/20 0.39
AR P10275 1/20 0.39
CHEK2 O96017 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
LCK P06239 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13617388 0.88 MAOB (0.46) MAOBEPHX2HDAC6VNN1ERN1
Benzene SCHEMBL27710673 0.85 MAOB (0.47) MAOBEPHX2HDAC6VNN1ERN1
SCHEMBL16121258 0.84 ACE2 (0.53) EPHX2
SCHEMBL403117 0.82 PDE3B (0.43) MAOBEPHX2HDAC6VNN1AR
SCHEMBL16380698 0.82 SLC6A2 (0.54) MAOBEPHX2HDAC6ARSLC6A2
SCHEMBL16140748 0.82 PKM (0.56) MAOBEPHX2HDAC6HSP90AA1HSP90AB1
SCHEMBL2709797 0.81 AR (0.45) MAOBVNN1ERN1PARP1PDK2
Hydrochloric Acid SCHEMBL27741712 0.79 AR (0.44) MAOBVNN1ERN1PARP1PDK2
SCHEMBL16140755 0.79 GSK3B (0.54) EPHX2HDAC6HSP90AA1HSP90AB1
SCHEMBL2777362 0.79 DDR1 (0.51) OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014206344-A1 FUSED TRICYCLIC AMIDE COMPOUNDS AS MULTIPLE KINASE INHIBITORS BEIGENE, LTD. (GB) 2014-12-31 WO disclosed