SCHEMBL16408530

SCHEMBL16408530

COC(=O)CCN1CCC[C@H]2C[C@@H]1c1cc(-c3ccc(C(F)(F)F)cc3)ccc12

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.69
TMEM97 Q5BJF2 3/20 0.69
HRH3 Q9Y5N1 3/20 0.42
TACR1 P25103 1/20 0.40
MGLL Q99685 1/20 0.38
BRD4 O60885 1/20 0.37
BRD2 P25440 1/20 0.37
BRD3 Q15059 1/20 0.37
KDM1A O60341 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CHRM3 P20309 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18100596 1.00 SIGMAR1 (0.69) SIGMAR1TMEM97HRH3TACR1MGLL
SCHEMBL21499080 1.00 SIGMAR1 (0.69) SIGMAR1TMEM97HRH3TACR1MGLL
SCHEMBL18099328 0.88 SIGMAR1 (0.52) SIGMAR1TMEM97HRH3
SCHEMBL18099332 0.85 SIGMAR1 (0.55) SIGMAR1TMEM97HRH3CHRM3
SCHEMBL16408535 0.85 SIGMAR1 (0.55) SIGMAR1TMEM97HRH3CHRM3
SCHEMBL18100571 0.85 SIGMAR1 (0.55) SIGMAR1TMEM97HRH3CHRM3
SCHEMBL16408637 0.85 SIGMAR1 (0.55) SIGMAR1TMEM97HRH3CHRM3
SCHEMBL21499079 0.82 SIGMAR1 (1.00) SIGMAR1TMEM97
SCHEMBL16408529 0.82 SIGMAR1 (1.00) SIGMAR1TMEM97
SCHEMBL21870943 0.82 SIGMAR1 (1.00) SIGMAR1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015009742-A2 COMPOUNDS AND METHODS FOR TREATING CANCER, NEUROLOGICAL DISORDERS, ETHANOL WITHDRAWAL, ANXIETY, DEPRESSION, AND NEUROPATHIC PAIN BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-01-22 WO disclosed