SCHEMBL16420396

SCHEMBL16420396

CC1CCc2c(Cl)ccnc21

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.39
HTR2A P28223 1/20 0.39
HTR2B P41595 1/20 0.39
HRH2 P25021 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
NISCH Q9Y2I1 1/20 0.33
ADRA1A P35348 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18807211 1.00 HTR2C (0.39) HTR2CHTR2AHTR2BHRH2HRH3
SCHEMBL1424574 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL29532721 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL4123694 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL15267245 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL12583743 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL30666992 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL379328 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL17768626 0.78 HTR2A (0.39) HTR2CHTR2AHTR2BFNTAFNTB
SCHEMBL15267240 0.77 HTR2B (0.37) HTR2CHTR2AHTR2BFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116134035-B 3- (1H-imidazol-2-yl) -2,3,8 a-tetrahydroindol-5 (1H) -one derivatives useful as factor XIA inhibitors 詹森药业有限公司 2025-03-11 CN disclosed
US-12043614-B2 Salts of a Pim kinase inhibitor INCYTE CORPORATION (US) 2024-07-23 US disclosed
US-20180170907-A1 SALTS OF A PIM KINASE INHIBITOR INCYTE CORPORATION 2018-06-21 US disclosed
US-9862705-B2 Salts of a pim kinase inhibitor INCYTE CORPORATION (US) 2018-01-09 US disclosed
US-20170121310-A1 SALTS OF A PIM KINASE INHIBITOR INCYTE CORPORATION 2017-05-04 US disclosed
EP-2185541-B1 Substituted phenylenediamines as inhibitors of the interaction between MDM2 and p53 JANSSEN PHARMACEUTICA NV (BE) 2015-01-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180170907-A1 SALTS OF A PIM KINASE INHIBITOR PIM1, PIM3, PIM2 HTR2C 3112/4885HTR2A 4423/4885HTR2B 4040/4885
US-20170121310-A1 SALTS OF A PIM KINASE INHIBITOR PIM1, PIM3, PIM2 HTR2C 3112/4885HTR2A 4423/4885HTR2B 4040/4885
US-12043614-B2 Salts of a Pim kinase inhibitor PIM1, PIM3, PIM2 HTR2C 3112/4885HTR2A 4423/4885HTR2B 4040/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.