SCHEMBL379328

SCHEMBL379328

OC1CCc2c(Cl)ccnc21

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
EPAS1 Q99814 1/20 0.37
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
P2RX7 Q99572 14/20 0.33
ACHE P22303 1/20 0.33
OPRL1 P41146 2/20 0.32
KCNH2 Q12809 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29532721 1.00 HTR2A (0.39) HTR2AHTR2CHTR2BEPAS1FNTA
SCHEMBL15267245 1.00 HTR2A (0.39) HTR2AHTR2CHTR2BEPAS1FNTA
SCHEMBL1424574 1.00 HTR2A (0.39) HTR2AHTR2CHTR2BEPAS1FNTA
SCHEMBL30666726 0.89 ACHE (0.43) HTR2AHTR2CHTR2BFNTAFNTB
SCHEMBL14884984 0.88 ACHE (0.39) HTR2AHTR2CHTR2BFNTAFNTB
SCHEMBL30667065 0.88 ACHE (0.39) HTR2AHTR2CHTR2BFNTAFNTB
SCHEMBL13270953 0.78 HTR2A (0.39) HTR2AHTR2CHTR2BEPAS1P2RX7
SCHEMBL12583743 0.78 HTR2A (0.39) HTR2AHTR2CHTR2BFNTAFNTB
SCHEMBL8263257 0.78 HTR2A (0.39) HTR2AHTR2CHTR2BEPAS1
SCHEMBL17768626 0.78 HTR2A (0.39) HTR2AHTR2CHTR2BFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 109 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250019366-A1 SALTS OF A PIM KINASE INHIBITOR INCYTE CORPORATION 2025-01-16 US claimed
CN-114380798-A Salts of Pim kinase inhibitors 因赛特公司 2022-04-22 CN claimed
US-20210155605-A1 SALTS OF A PIM KINASE INHIBITOR INCYTE CORPORATION 2021-05-27 US claimed
US-20170121310-A1 SALTS OF A PIM KINASE INHIBITOR INCYTE CORPORATION 2017-05-04 US claimed
EP-4695240-A2 CYCLIC VINYL SULFONE WRN INHIBITORS Nimbus Wadjet, Inc. (US) 2026-02-18 EP disclosed
US-20260035379-A1 BICYCLIC PYRIDINE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2026-02-05 US disclosed
US-12534475-B2 Bicyclic pyridine derivative Sumitomo Pharma Co., Ltd. (JP) 2026-01-27 US disclosed
US-20250066357-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2025-02-27 US disclosed
US-20250019366-A1 SALTS OF A PIM KINASE INHIBITOR INCYTE CORPORATION 2025-01-16 US disclosed
US-12187721-B2 Protein tyrosine phosphatase inhibitors ARRAY BIOPHARMA INC. (US) 2025-01-07 US disclosed
WO-2024215923-A2 CYCLIC VINYL SULFONE WRN INHIBITORS NIMBUS WADJET, INC. (US) 2024-10-17 WO disclosed
US-12077546-B2 Bicyclic pyridine derivative Sumitomo Pharma Co., Ltd. (JP) 2024-09-03 US disclosed
EP-2203447-A1 INHIBITORS OF THE INTERACTION BETWEEN MDM2 AND P53 Janssen Pharmaceutica, N.V. (BE) 2010-07-07 EP disclosed
US-20100168065-A1 QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-07-01 US disclosed
EP-2134691-A1 QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS Janssen Pharmaceutica, N.V. (BE) 2009-12-23 EP disclosed
WO-2009118384-A1 QUINAZOLINONE DERIVATIVES AS TUBULIN POLYMERIZATION INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2009-10-01 WO disclosed
WO-2009037308-A1 INHIBITORS OF THE INTERACTION BETWEEN MDM2 AND P53 JANSSEN PHARMACEUTICA NV (BE) 2009-03-26 WO disclosed
WO-2009037343-A1 INHIBITORS OF THE INTERACTION BETWEEN MDM2 AND P53 JANSSEN PHARMACEUTICA NV (BE) 2009-03-26 WO disclosed
WO-2009019274-A1 SUBSTITUTED PHENYLENEDIAMINES AS INHIBITORS OF THE INTERACTION BETWEEN MDM2 AND P53 JANSSEN PHARMACEUTICA NV (BE) 2009-02-12 WO disclosed
WO-2008107478-A1 QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260035379-A1 BICYCLIC PYRIDINE DERIVATIVE CBR1, CBR3, CYP2B6 HTR2A 642/4885HTR2C 138/4885HTR2B 453/4885
US-20250066357-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS PPM1A, PPM1F, PPP5C HTR2A 4536/4885HTR2C 4347/4885HTR2B 4580/4885
US-12187721-B2 Protein tyrosine phosphatase inhibitors PPM1A, PTP4A1, PPP5C HTR2A 4423/4885HTR2C 4302/4885HTR2B 4425/4885
US-12077546-B2 Bicyclic pyridine derivative CBR1, CBR3, CYB5R3 HTR2A 1075/4885HTR2C 428/4885HTR2B 304/4885
US-20210155605-A1 SALTS OF A PIM KINASE INHIBITOR PIM1, PIM3, PIM2 HTR2A 4423/4885HTR2C 3112/4885HTR2B 4040/4885
US-20100168065-A1 QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS PARP1, PARP11, PARP3 HTR2A 1515/4885HTR2C 2169/4885HTR2B 1959/4885
US-20250019366-A1 SALTS OF A PIM KINASE INHIBITOR PIM1, PIM2, PIM3 HTR2A 4403/4885HTR2C 3100/4885HTR2B 4003/4885
US-20170121310-A1 SALTS OF A PIM KINASE INHIBITOR PIM1, PIM3, PIM2 HTR2A 4423/4885HTR2C 3112/4885HTR2B 4040/4885
US-12534475-B2 Bicyclic pyridine derivative CBR1, CYP2B6, CBR3 HTR2A 407/4885HTR2C 63/4885HTR2B 296/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.