SCHEMBL16442162

SCHEMBL16442162

COc1cc(-c2cc3cc(OCCCN4CCC(O)CC4)ccc3n2CC(C)=O)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.45
HRH2 P25021 3/20 0.45
HRH1 P35367 3/20 0.45
SIGMAR1 Q99720 3/20 0.41
MAOB P27338 1/20 0.41
PAX8 Q06710 1/20 0.41
SLC6A4 P31645 1/20 0.40
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16424320 0.89 AVPR1B (0.49) HRH3
SCHEMBL16423585 0.85 AVPR1B (0.47) HRH3HRH2HRH1
SCHEMBL16445077 0.81 AVPR1B (0.48) HRH3HRH2HRH1
SCHEMBL16423839 0.81 AVPR1B (0.57)
SCHEMBL16424040 0.76 AVPR1B (0.55) HRH3KCNH2
SCHEMBL16442153 0.76 BACE1 (0.39)
SCHEMBL16423675 0.75 AVPR1B (0.59)
SCHEMBL16423778 0.74 AVPR1B (0.47)
SCHEMBL16423724 0.73 AVPR1B (0.45)
SCHEMBL6857474 0.72 AVPR1B (0.45) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2832722-A1 FUSED AZOLE DERIVATIVE Taisho Pharmaceutical Co., Ltd. (JP) 2015-02-04 EP disclosed