SCHEMBL16456992

SCHEMBL16456992

CC(C)N1CCC(c2nc3cc(-c4cccc(F)c4Cl)nc(N4CCCC(Nc5ccc(C(=O)C(F)(F)F)c(N)n5)C4)n3n2)CC1

nearest known ligand 0.31

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
WNT1 P04628 1/20 0.31
DYRK1A Q13627 1/20 0.31
EGFR P00533 1/20 0.31
LCK P06239 1/20 0.31
JAK3 P52333 1/20 0.31
BTK Q06187 1/20 0.31
IL1B P01584 1/20 0.30
BMPR1B O00238 1/20 0.30
BMPR1A P36894 1/20 0.30
TGFBR1 P36897 1/20 0.30
ACVRL1 P37023 1/20 0.30
ACVR1 Q04771 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1120117 0.90 MAPK14 (0.32) EGFRLCKJAK3BTKIL1B
SCHEMBL1962713 0.90 BMPR1B (0.34) EGFRLCKJAK3BTKIL1B
SCHEMBL1962175 0.90 GSK3B (0.35) EGFRLCKJAK3BTKIL1B
SCHEMBL1960445 0.82 ACKR3 (0.36) EGFRLCKJAK3BTKBMPR1B
SCHEMBL8003442 0.81 GSK3B (0.37) EGFRLCKJAK3BTK
SCHEMBL1119579 0.80 BMPR1B (0.32) EGFRLCKJAK3BTKBMPR1B
SCHEMBL12579257 0.80 BMPR1B (0.31) IL1BBMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL1962515 0.77 DPP4 (0.34)
SCHEMBL1120223 0.77 DPP4 (0.34)
SCHEMBL1119497 0.74 MAPK14 (0.34) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2280976-B1 SUBSTITUTED IMIDAZO- AND TRIAZOLOPYRIMIDINES, IMIDAZO- AND PYRAZOLOPYRAZINES AND IMIDAZOTRIAZINES AS GSK3BETA-INHIBITORS BAYER IP GMBH (DE) 2014-01-01 EP disclosed