SCHEMBL16457900

SCHEMBL16457900

c1cnc2[nH]ncc2c1.c1cnnnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.42
AXL P30530 1/20 0.42
HSP90AA1 P07900 2/20 0.41
IDO1 P14902 1/20 0.41
CDK2 P24941 1/20 0.41
DAO P14920 1/20 0.39
PIM1 P11309 1/20 0.38
PIM3 Q86V86 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
FGFR1 P11362 1/20 0.37
IKBKE Q14164 1/20 0.36
TBK1 Q9UHD2 1/20 0.36
NOS1 P29475 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 2/20 0.36
PARP1 P09874 1/20 0.36
PRKCI P41743 1/20 0.36
PDE4B Q07343 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7679 0.90
SCHEMBL29365139 0.90
SCHEMBL23159915 0.88 NUDT1 (0.48) NUDT1AXLHSP90AA1IDO1CDK2
Hydrochloric Acid SCHEMBL16296100 0.88 NUDT1 (0.48) NUDT1AXLHSP90AA1IDO1CDK2
Urea SCHEMBL28419880 0.79 FLT3 (0.49) NUDT1AXLHSP90AA1IDO1CDK2
Dipyridyl SCHEMBL28565857 0.79 KDM4E (0.52) HSP90AA1IDO1CDK2PIM1TDP1
SCHEMBL5025757 0.77 CDK2 (0.50) NUDT1AXLHSP90AA1IDO1CDK2
SCHEMBL11903658 0.77 CDK2 (0.50) NUDT1AXLHSP90AA1IDO1CDK2
Fumaric Acid SCHEMBL10591225 0.75 KDM4E (0.49) NUDT1AXLDAOPIM1PIM3
Maleic Acid SCHEMBL10591220 0.75 KDM4E (0.49) NUDT1AXLDAOPIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2682394-A1 1H-pyrazolo[3,4-b]pyridin-triazine derivatives and their use for the treatment or the prevention of cardiovascular diseases Bayer Intellectual Property GmbH (DE) 2014-01-08 EP disclosed