SCHEMBL16458014

SCHEMBL16458014

CC(CCNC(=O)C(c1ccc(CN2N=C(c3ccccc3)OCC2=O)cc1)C1CCCC1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PTGS2 P35354 6/20 0.38
PTGES O14684 2/20 0.37
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16457356 0.95 TP53 (0.43) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL517018 0.95 TP53 (0.43) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL1725285 0.94 TP53 (0.42) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL1178266 0.87 BDKRB2 (0.41) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL517315 0.87 TP53 (0.46) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL516846 0.87 TP53 (0.40) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL518071 0.86 TP53 (0.45) TP53CYP1A2CYP3A4CYP2D6TSHR
Bicarbonate SCHEMBL1079990 0.86 BDKRB2 (0.43) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL517236 0.86 TDP1 (0.43) TP53CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL516987 0.86 TP53 (0.41) TP53CYP1A2CYP3A4CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406215-B1 OXO-HETEROCYCLICALLY SUBSTITUTED ALKYL CARBOXYLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2014-04-16 EP disclosed