SCHEMBL16460465

SCHEMBL16460465

NCC(c1ccc(F)nc1)N1CCC(F)(F)CC1

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 16/20 0.54
RPS6KB1 P23443 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12701152 0.86 P2RX7 (0.42) P2RX7RPS6KB1
SCHEMBL12701169 0.85 RPS6KB1 (0.52) P2RX7RPS6KB1
SCHEMBL16461777 0.85 P2RX7 (0.53) P2RX7RPS6KB1
SCHEMBL16395576 0.85 RPS6KB1 (0.52) P2RX7RPS6KB1
SCHEMBL16395501 0.85 RPS6KB1 (0.52) P2RX7RPS6KB1
SCHEMBL16460147 0.84 P2RX7 (0.57) P2RX7RPS6KB1
SCHEMBL12701210 0.83 P2RX7 (0.57) P2RX7RPS6KB1
SCHEMBL12701316 0.81 P2RX7 (0.41) P2RX7
SCHEMBL16460909 0.81 P2RX7 (0.48) P2RX7RPS6KB1
SCHEMBL12701124 0.80 P2RX7 (0.53) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190307766-A1 CYCLIC AMINES MINDIMMUNE THERAPEUTICS, INC. 2019-10-10 US disclosed
US-20190307766-A1 CYCLIC AMINES MINDIMMUNE THERAPEUTICS, INC. 2019-10-10 US disclosed
EP-3536689-A1 2-(CYCLIC AMINEETHYL)BENZAMIDE DERIVATIVES AS P2X7 INHIBITORS MindImmune Therapeutics, Inc. (US) 2019-09-11 EP disclosed
EP-2906549-B1 N-(2-(CYCLIC AMINE)ETHYL)BENZAMIDE DERIVATIVES AS P2X7 INHIBITORS MINDIMMUNE THERAPEUTICS INC (US) 2019-04-17 EP disclosed
US-10124010-B2 Cyclic amines MINDIMMUNE THERAPEUTICS, INC. (US) 2018-11-13 US disclosed
US-20180177793-A1 CYCLIC AMINES MINDIMMUNE THERAPEUTICS, INC. 2018-06-28 US disclosed
US-20180177793-A1 CYCLIC AMINES MINDIMMUNE THERAPEUTICS, INC. 2018-06-28 US disclosed
US-20180177793-A1 CYCLIC AMINES MINDIMMUNE THERAPEUTICS, INC. 2018-06-28 US disclosed
US-9861639-B2 Cyclic amines H. LUNDBECK A/S (DK) 2018-01-09 US disclosed
US-9861639-B2 Cyclic amines H. LUNDBECK A/S (DK) 2018-01-09 US disclosed
US-20150306114-A1 Cyclic Amines MINDIMMUNE THERAPEUTICS, INC. 2015-10-29 US disclosed
EP-2906549-A2 CYCLIC AMINES H. Lundbeck A/S (DK) 2015-08-19 EP disclosed
US-9108938-B2 Cyclic amines H. LUNDBECK A/S (DK) 2015-08-18 US disclosed
US-9108938-B2 Cyclic amines H. LUNDBECK A/S (DK) 2015-08-18 US disclosed
US-9108938-B2 Cyclic amines H. LUNDBECK A/S (DK) 2015-08-18 US disclosed
US-20140107335-A1 Cyclic Amines H. LUNDBECK A/S (DK) 2014-04-17 US disclosed
US-20140107335-A1 Cyclic Amines H. LUNDBECK A/S (DK) 2014-04-17 US disclosed
WO-2014057080-A2 CYCLIC AMINES H. LUNDBECK A/S (DK) 2014-04-17 WO disclosed
US-20140107335-A1 Cyclic Amines H. LUNDBECK A/S (DK) 2014-04-17 US disclosed
WO-2014057080-A2 CYCLIC AMINES H. LUNDBECK A/S (DK) 2014-04-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150306114-A1 Cyclic Amines P2RX7, ADORA2A, P2RX2 P2RX7 1/4885RPS6KB1 2290/4885
US-20190307766-A1 CYCLIC AMINES P2RX7, ADORA2A, P2RX2 P2RX7 1/4885RPS6KB1 2290/4885
US-20140107335-A1 Cyclic Amines P2RX7, ADORA2A, P2RX2 P2RX7 1/4885RPS6KB1 2290/4885
US-10124010-B2 Cyclic amines P2RX7, ADORA2A, P2RX2 P2RX7 1/4885RPS6KB1 2290/4885
US-20180177793-A1 CYCLIC AMINES P2RX7, ADORA2A, P2RX2 P2RX7 1/4885RPS6KB1 2290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.