SCHEMBL16464883

SCHEMBL16464883

CCNC(=O)C1Cc2cccnc2N1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHIA Q9BZP6 1/20 0.44
LMNA P02545 2/20 0.41
MTNR1A P48039 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HTR7 P34969 1/20 0.38
CYP46A1 Q9Y6A2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17094786 0.85 CHIA (0.41) CHIALMNAKDM4E
SCHEMBL16466327 0.83 KDM4E (0.43) CHIALMNAMTNR1AALDH1A1KDM4E
SCHEMBL16466326 0.83 KDM4E (0.43) CHIALMNAMTNR1AALDH1A1KDM4E
SCHEMBL16462753 0.83 XIAP (0.47) CHIALMNAALDH1A1KDM4ECYP1A2
SCHEMBL16466185 0.81 KDM4E (0.39) CHIAMTNR1AKDM4E
SCHEMBL16465007 0.80 NR1D1 (0.42) ALDH1A1KDM4E
SCHEMBL16465263 0.78 XIAP (0.60)
SCHEMBL16464394 0.78 XIAP (0.60)
SCHEMBL16465261 0.78 XIAP (0.60)
SCHEMBL16466120 0.77 XIAP (0.45) LMNAALDH1A1KDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906559-A1 AZAINDOLINES F. Hoffmann-La Roche AG (CH) 2015-08-19 EP disclosed
WO-2014056871-A1 AZAINDOLINES F. HOFFMANN-LA ROCHE AG (CH) 2014-04-17 WO disclosed