SCHEMBL16465327

SCHEMBL16465327

NC(=O)c1cnc(N)nc1-c1ccccc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 5/20 0.52
DBF4 Q9UBU7 1/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
PARP1 P09874 1/20 0.48
ADORA2A P29274 2/20 0.47
EPAS1 Q99814 1/20 0.42
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
PRKD3 O94806 1/20 0.42
MAPK9 P45984 1/20 0.42
MAPKAPK2 P49137 1/20 0.42
MAPK10 P53779 1/20 0.42
ROCK1 Q13464 1/20 0.42
ACVR2B Q13705 1/20 0.42
MYLK Q15746 1/20 0.42
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
PRKD2 Q9BZL6 1/20 0.42
NLK Q9UBE8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29058641 0.88 NPC1 (0.52) CDC7DBF4NPC1RAB9AADORA2A
SCHEMBL30395416 0.88 NPC1 (0.52) CDC7DBF4NPC1RAB9AADORA2A
SCHEMBL29058668 0.83 KMT2A (0.43) CDC7DBF4NPC1RAB9AADORA2A
SCHEMBL30395322 0.83 KMT2A (0.43) CDC7DBF4NPC1RAB9AADORA2A
SCHEMBL15648676 0.79 ADORA2A (0.56) CDC7DBF4NPC1ADORA2AALOX5AP
SCHEMBL4560200 0.78 CDC7 (0.56) CDC7PARP1ADORA2AADORA1JAK2
SCHEMBL18351966 0.78 ADORA1 (0.51) CDC7PARP1ADORA2AMAPK10ADORA1
SCHEMBL15622225 0.77 SIRT1 (0.52) CDC7ADORA2AEPAS1ADORA1KDM4E
SCHEMBL15621842 0.77 CDC7 (0.42) CDC7
SCHEMBL4183400 0.76 CDC7 (0.72) CDC7PRKD3MAPK9ROCK1PRKD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903970-A2 SUBSTITUTED PYRIMIDINYL KINASE INHIBITORS Portola Pharmaceuticals, Inc. (US) 2015-08-12 EP claimed
WO-2014058921-A2 SUBSTITUTED PYRIMIDINYL KINASE INHIBITORS PORTOLA PHARMACEUTICALS, INC. (US) 2014-04-17 WO claimed