SCHEMBL16465757

SCHEMBL16465757

COC(=O)C(=CN(O)C(C)C(C)C)C(=O)c1cc(Br)c(OC)cc1OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
CYP3A4 P08684 1/20 0.35
KDM4E B2RXH2 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RECQL P46063 1/20 0.33
PAX8 Q06710 1/20 0.32
ALDH1A1 P00352 2/20 0.32
TNFRSF1A P19438 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
LCK P06239 1/20 0.31
FYN P06241 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16465755 1.00 ABCB1 (0.36) ABCB1MAPTHPGDCYP3A4KDM4E
SCHEMBL16462423 0.89 ABCB1 (0.37) ABCB1CYP3A4KDM4ENPSR1RECQL
SCHEMBL16462426 0.89 ABCB1 (0.37) ABCB1CYP3A4KDM4ENPSR1RECQL
SCHEMBL16461663 0.83 MAPT (0.40) ABCB1MAPTHPGDCYP3A4KDM4E
SCHEMBL16461664 0.83 MAPT (0.40) ABCB1MAPTHPGDCYP3A4KDM4E
SCHEMBL16462243 0.75 CYP3A4 (0.35) CYP3A4KDM4ENPSR1PAX8LMNA
SCHEMBL16462241 0.75 CYP3A4 (0.35) CYP3A4KDM4ENPSR1PAX8LMNA
SCHEMBL18240186 0.75 MAPT (0.34) ABCB1MAPTHPGDCYP3A4KDM4E
SCHEMBL18240184 0.75 MAPT (0.34) ABCB1MAPTHPGDCYP3A4KDM4E
SCHEMBL18627854 0.75 MAPT (0.34) ABCB1MAPTHPGDCYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906540-A1 AN IMPROVED PRODUCTION METHOD AND NEW INTERMEDIATES OF SYNTHESIS OF ELVITEGRAVIR Zentiva K.S. (CZ) 2015-08-19 EP disclosed
WO-2014056465-A1 AN IMPROVED PRODUCTION METHOD AND NEW INTERMEDIATES OF SYNTHESIS OF ELVITEGRAVIR ZENTIVA, K.S. (CZ) 2014-04-17 WO disclosed