SCHEMBL16472002

SCHEMBL16472002

CCCS/C(N)=N\Cc1cccc(NC(=O)c2cnc(N(C)C)cn2)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 9/20 0.40
SIRT1 Q96EB6 9/20 0.40
SIRT3 Q9NTG7 9/20 0.40
AURKA O14965 2/20 0.40
RPS6KB1 P23443 2/20 0.40
AURKB Q96GD4 2/20 0.40
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
BACE1 P56817 4/20 0.39
PARP1 P09874 1/20 0.39
HRH4 Q9H3N8 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
ACKR3 P25106 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10193147 0.85 BACE1 (0.47) SIRT2SIRT1SIRT3BACE1
SCHEMBL10155847 0.81 BACE1 (0.59) BACE1
SCHEMBL10193014 0.80 BACE1 (0.46) SIRT2SIRT1SIRT3BACE1HRH4
SCHEMBL10192928 0.78 BACE1 (0.46) SIRT2SIRT1SIRT3ALDH1A1BACE1
SCHEMBL10193824 0.78 BACE1 (0.45) BACE1HRH4HRH3
SCHEMBL10193935 0.78 BACE1 (0.45) SIRT2SIRT1SIRT3BACE1HRH4
SCHEMBL10193785 0.77 BACE1 (0.48) SIRT2SIRT1SIRT3BACE1
SCHEMBL10155870 0.76 BACE1 (0.57) BACE1
SCHEMBL10193222 0.75 ALDH1A1 (0.51) AURKARPS6KB1ALDH1A1TDP1BACE1
SCHEMBL10192932 0.75 BACE1 (0.46) SIRT2SIRT1SIRT3ALDH1A1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942105-B1 AMINODIHYDROTHIAZINE DERIVATIVE SHIONOGI & CO (JP) 2014-04-16 EP disclosed