SCHEMBL1647235

SCHEMBL1647235

COc1cccc(CN(C)C(=O)c2cn(CCCO)c3cc(-c4cn[nH]c4)ccc23)c1

nearest known ligand 0.84

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 16/20 0.84
ROCK1 Q13464 15/20 0.84
CYP2C9 P11712 1/20 0.53
CDC42BPA Q5VT25 1/20 0.53
PRKACA P17612 2/20 0.52
PRKACG P22612 2/20 0.52
PRKACB P22694 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647659 0.91 ROCK1 (1.00) ROCK2ROCK1CYP2C9CDC42BPAPRKACA
SCHEMBL1647662 0.88 ROCK1 (1.00) ROCK2ROCK1CYP2C9CDC42BPAPRKACA
SCHEMBL1648105 0.88 ROCK2 (0.83) ROCK2ROCK1
SCHEMBL12779542 0.85 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647861 0.83 ROCK1 (0.85) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648742 0.81 ROCK2 (1.00) ROCK2ROCK1CYP2C9CDC42BPAPRKACA
SCHEMBL1649576 0.80 ROCK1 (0.91) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647286 0.79 ROCK1 (1.00) ROCK2ROCK1CYP2C9CDC42BPAPRKACA
SCHEMBL1648804 0.79 ROCK2 (1.00) ROCK2ROCK1CYP2C9CDC42BPAPRKACA
SCHEMBL1647243 0.78 ROCK2 (1.00) ROCK2ROCK1CYP2C9CDC42BPAPRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed