SCHEMBL16473589

SCHEMBL16473589

Nc1ncc(-c2nc(N3CCOC[C@@H]3N)c3ncn(CC(F)(F)F)c3n2)cn1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.48
MTOR P42345 7/20 0.46
PIK3CD O00329 4/20 0.46
PIK3CB P42338 4/20 0.46
PIK3R1 P27986 4/20 0.46
PIK3CG P48736 3/20 0.46
HDAC1 Q13547 3/20 0.46
RPTOR Q8N122 4/20 0.44
MLST8 Q9BVC4 4/20 0.44
RICTOR Q6R327 3/20 0.44
MAPKAP1 Q9BPZ7 3/20 0.44
PIK3C3 Q8NEB9 1/20 0.43
ATR Q13535 1/20 0.43
MAP3K12 Q12852 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL336266 0.90 PIK3CA (0.56) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL336979 0.84 PIK3CA (0.67) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL799640 0.80 PIK3CA (0.62) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL13674676 0.78 PIK3CA (0.60) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL336390 0.76 PIK3CA (0.57) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL799327 0.74 MTOR (0.52) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL337181 0.72 PIK3CA (0.62) PIK3CAMTORPIK3CDPIK3CBPIK3R1
Bicarbonate SCHEMBL13674675 0.72 HDAC1 (0.53) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL336204 0.71 PIK3CA (0.67) PIK3CAMTORPIK3CDPIK3CBPIK3R1
SCHEMBL336242 0.71 MTOR (0.47) PIK3CAMTORPIK3CDRPTORMLST8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2336132-B1 MORPHOLINOPURINE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2014-01-01 EP disclosed