SCHEMBL16474292

SCHEMBL16474292

F[C@@H]1CCN(c2ccccn2)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 1/20 0.51
GRIN2D O15399 1/20 0.47
GRIN3B O60391 1/20 0.47
GRIN1 Q05586 1/20 0.47
GRIN2A Q12879 1/20 0.47
GRIN2B Q13224 1/20 0.47
GRIN2C Q14957 1/20 0.47
GRIN3A Q8TCU5 1/20 0.47
USP30 Q70CQ3 1/20 0.47
KDM4E B2RXH2 2/20 0.46
GRM1 Q13255 1/20 0.46
GPR119 Q8TDV5 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA4 P22748 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18833378 0.87 PLD1 (0.52) PLD1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3154404 0.84 HRH4 (0.51) PLD1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3658830 0.84 HRH4 (0.51) PLD1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3153901 0.84 HRH4 (0.51) PLD1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL28170653 0.83 MAP4K4 (0.49) PLD1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL31549832 0.83 MAP4K4 (0.49) PLD1GRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL1402090 0.83 HRH4 (0.50) PLD1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL31441374 0.83 PLD1 (0.53) PLD1KDM4EGPR119SMN1; SMN2HSD17B10
Hydrochloric Acid SCHEMBL1402092 0.83 HRH4 (0.50) PLD1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL23875675 0.81 GRM1 (0.51) PLD1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523954-B1 1H-[1,2,3]TRIAZOLO[4,5-C]PYRIDINE-4- CARBONITRILE DERIVATIVES AS CATHEPSIN S INHIBITORS MERCK SHARP & DOHME (NL) 2014-04-16 EP disclosed