SCHEMBL28170653

SCHEMBL28170653

FC(F)(F)C1CCN(c2ccccn2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.49
DPP4 P27487 1/20 0.46
DPP8 Q6V1X1 1/20 0.46
DPP9 Q86TI2 1/20 0.46
DPP7 Q9UHL4 1/20 0.46
PLD1 Q13393 1/20 0.46
GRM1 Q13255 2/20 0.45
HTT P42858 1/20 0.45
AVPR1A P37288 1/20 0.44
PDE10A Q9Y233 1/20 0.44
USP30 Q70CQ3 1/20 0.43
GPR119 Q8TDV5 2/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
GRIN1 Q05586 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43
GRIN2C Q14957 1/20 0.43
GRIN3A Q8TCU5 1/20 0.43
CA12 O43570 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31549832 1.00 MAP4K4 (0.49) MAP4K4DPP4DPP8DPP9DPP7
SCHEMBL30641568 0.90 PLD1 (0.53) PLD1HTTAVPR1APDE10AGPR119
SCHEMBL30641563 0.90 PLD1 (0.53) PLD1HTTAVPR1APDE10AGPR119
SCHEMBL16543107 0.84 GRM1 (0.57) PLD1GRM1AVPR1AUSP30GPR119
SCHEMBL16474292 0.83 PLD1 (0.51) PLD1GRM1AVPR1AUSP30GPR119
SCHEMBL17619606 0.81 GPR119 (0.52) PLD1GRM1HTTAVPR1AGPR119
SCHEMBL28136848 0.80 KDM4E (0.45) MAP4K4DPP4DPP8DPP9DPP7
SCHEMBL16785630 0.78 MAP4K4 (0.46) MAP4K4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL896038 0.76 DPP4 (0.51) DPP4DPP8DPP9DPP7GRM1
SCHEMBL25253230 0.76 MAP4K4 (0.50) MAP4K4PDE10AGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107207496-A Substituted bridged ring urea analogs as sirtuin modulators 葛兰素史密斯克莱有限责任公司 2017-09-26 CN disclosed