SCHEMBL16474651

SCHEMBL16474651

CCCC(CCC)c1nc2cc(-c3ccc(Cl)cc3Cl)nc(NCCNc3ccc(C(=O)CC)c(N)n3)n2n1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.34
ALPL P05186 5/20 0.34
CRHR1 P34998 4/20 0.34
GSK3B P49841 4/20 0.33
GSK3A P49840 2/20 0.33
CNR1 P21554 2/20 0.33
CDK1 P06493 1/20 0.31
POLB P06746 1/20 0.31
THRB P10828 1/20 0.31
RECQL P46063 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
ALPG P10696 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1963687 0.82 DPP4 (0.36) DPP4ALPLCRHR1GSK3BGSK3A
SCHEMBL12680892 0.75 GSK3B (0.36) DPP4ALPLGSK3BGSK3ACNR1
SCHEMBL12680888 0.74 ADORA2A (0.40) DPP4GSK3BGSK3ACNR1DPP8
SCHEMBL12680846 0.73 ALPL (0.37) DPP4ALPLGSK3BGSK3ACNR1
SCHEMBL1119573 0.73 DPP4 (0.36) DPP4GSK3BGSK3ACDK1
SCHEMBL1960159 0.72 GSK3B (0.39) DPP4ALPLGSK3BGSK3ACNR1
SCHEMBL1964817 0.72 GSK3B (0.33) DPP4GSK3BGSK3A
SCHEMBL9105999 0.72 GSK3B (0.39) DPP4ALPLGSK3BGSK3ACDK1
SCHEMBL12680862 0.71 GSK3B (0.36) ALPLGSK3BGSK3ACDK1ALPG
SCHEMBL12680864 0.71 GSK3B (0.38) DPP4ALPLGSK3BGSK3ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2280976-B1 SUBSTITUTED IMIDAZO- AND TRIAZOLOPYRIMIDINES, IMIDAZO- AND PYRAZOLOPYRAZINES AND IMIDAZOTRIAZINES AS GSK3BETA-INHIBITORS BAYER IP GMBH (DE) 2014-01-01 EP disclosed