SCHEMBL16477207

SCHEMBL16477207

Brc1ccc2c3c([nH]c2c1)CCCNC3

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.53
TAAR1 Q96RJ0 1/20 0.49
HSD17B10 Q99714 1/20 0.48
MCHR1 Q99705 3/20 0.44
NISCH Q9Y2I1 2/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
HTR7 P34969 1/20 0.43
RAD52 P43351 1/20 0.40
KMT2A Q03164 1/20 0.40
PARP1 P09874 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HTR5A P47898 1/20 0.40
NR2E1 Q9Y466 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
PNMT P11086 1/20 0.39
ASIC3 Q9UHC3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18345852 0.91 TAAR1 (0.59) MAPTTAAR1HSD17B10NISCHADRA2A
SCHEMBL6627508 0.82 MAPT (0.75) MAPTHSD17B10KMT2AKDM4E
SCHEMBL1004931 0.82 MAPT (0.70) MAPTHSD17B10KMT2APARP1KDM4E
SCHEMBL3476066 0.81 NISCH (0.62) MAPTTAAR1HSD17B10NISCHADRA2A
SCHEMBL29773845 0.81 NISCH (0.62) MAPTTAAR1HSD17B10NISCHADRA2A
SCHEMBL12927815 0.81 MAPT (0.68) MAPTHSD17B10KMT2APARP1KDM4E
SCHEMBL411353 0.78 MAPT (0.64) MAPTTAAR1HSD17B10RAD52KMT2A
SCHEMBL620253 0.78 TAAR1 (0.78) TAAR1NISCHPARP1KDM4EHTR5A
Hydrochloric Acid SCHEMBL18345594 0.77 TAAR1 (0.62) MAPTTAAR1HSD17B10RAD52KMT2A
SCHEMBL10155124 0.73 PARP1 (0.56) MAPTTAAR1RAD52KMT2APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2448585-B1 AZINONE-SUBSTITUTED AZEPINO[B]INDOLE AND PYRIDO-PYRROLO-AZEPINE MCH-1 ANTAGONISTS, METHODS OF MAKING, AND USE THEREOF ALBANY MOLECULAR RES INC (US) 2014-01-01 EP disclosed