SCHEMBL16478136

SCHEMBL16478136

CC(C)N1Cc2cc(-c3ccc(C(C#N)CNC(=O)N(C(=O)O)C4CCCCC4)cc3)cnc2C1=O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.33
CTSK P43235 1/20 0.31
CTSC P53634 1/20 0.31
PDE3B Q13370 4/20 0.31
PDE3A Q14432 4/20 0.31
MAPK1 P28482 1/20 0.31
KCNH2 Q12809 2/20 0.31
PIK3CG P48736 4/20 0.30
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
BACE1 P56817 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290330 0.91 CTSC (0.38) ACACBCTSKCTSCPDE3BPDE3A
SCHEMBL16478361 0.86 CTSK (0.35) ACACBCTSKCTSCKCNH2PIK3CG
SCHEMBL16478214 0.83 F9 (0.38) ACACBCTSKCTSCPDE3BPDE3A
SCHEMBL16478162 0.81 KCNH2 (0.32) ACACBCTSKCTSCKCNH2PIK3CG
SCHEMBL16478134 0.79 PIK3CG (0.32) CTSKCTSCMAPK1PIK3CG
SCHEMBL16478104 0.78 JAK2 (0.34) ACACBCTSCROCK2ROCK1
SCHEMBL16478194 0.77 PDE4A (0.38) ACACBCTSCROCK2ROCK1
SCHEMBL16478066 0.76 ACACB (0.34) ACACBCTSKROCK2ROCK1
SCHEMBL16478221 0.74 CTSC (0.38) CTSKCTSCKCNH2ROCK2ROCK1
SCHEMBL16478103 0.74 CTSC (0.41) CTSKCTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011154677-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL] 1-AMINOCYCLOALK-1-YLCARBOXAMIDE COMPOUNDS - 760 ASTRAZENECA AB (SE) 2011-12-15 WO disclosed