SCHEMBL16478337

SCHEMBL16478337

CCS(=O)(=O)c1ccc(-c2ccc(CC(NC(=O)C3(NC(=O)O)CCCCC3)C(N)=O)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.52
ITGA4 P13612 15/20 0.52
ECE1 P42892 3/20 0.45
ITGB7 P26010 3/20 0.43
RORC P51449 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16478305 0.99 ITGB1 (0.51) ITGB1ITGA4ECE1ITGB7RORC
SCHEMBL298671 0.90 ITGB1 (0.44) ITGB1ITGA4ECE1ITGB7RORC
SCHEMBL16478312 0.86 ITGB1 (0.42) ITGB1ITGA4ECE1ITGB7
SCHEMBL16478311 0.86 ITGB1 (0.42) ITGB1ITGA4ECE1ITGB7
SCHEMBL299948 0.84 ITGB1 (0.42) ITGB1ITGA4ECE1ITGB7
SCHEMBL16478164 0.83 CTSC (0.54) ITGB1ITGA4
SCHEMBL16478181 0.81 ECE1 (0.43) ITGB1ITGA4ECE1ITGB7
SCHEMBL16478172 0.81 TACR2 (0.45) ITGB1ITGA4ECE1
SCHEMBL16478145 0.81 TACR2 (0.45) ITGB1ITGA4ECE1
SCHEMBL16478073 0.81 CTSC (0.53) ITGB1ITGA4ECE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011154677-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL] 1-AMINOCYCLOALK-1-YLCARBOXAMIDE COMPOUNDS - 760 ASTRAZENECA AB (SE) 2011-12-15 WO disclosed