SCHEMBL299948

SCHEMBL299948

CCCS(=O)(=O)c1ccc(-c2ccc(CC(NC(=O)C3(NC(=O)O)CCOCC3)C(N)=O)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 12/20 0.42
ITGA4 P13612 12/20 0.42
ITGB7 P26010 4/20 0.41
CTSC P53634 2/20 0.39
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA9 Q16790 2/20 0.38
TACR2 P21452 2/20 0.38
ECE1 P42892 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298671 0.94 ITGB1 (0.44) ITGB1ITGA4ITGB7CTSCTACR2
SCHEMBL16478305 0.85 ITGB1 (0.51) ITGB1ITGA4ITGB7ECE1
SCHEMBL16478337 0.84 ITGB1 (0.52) ITGB1ITGA4ITGB7ECE1
SCHEMBL299110 0.84 ALDH1A1 (0.51) ITGB1ITGA4TACR2
SCHEMBL289666 0.83 ALDH1A1 (0.46) ITGB1ITGA4CTSCTACR2
SCHEMBL298498 0.83 CTSC (0.59) ITGB1ITGA4ITGB7CTSCTACR2
SCHEMBL298999 0.83 CTSC (0.44) ITGB1ITGA4ITGB7CTSCTACR2
SCHEMBL298776 0.82 SMN1; SMN2 (0.44) ITGB1ITGA4CTSCTACR2
SCHEMBL2892835 0.81 ITGB1 (0.41) ITGB1ITGA4ITGB7CTSCTACR2
SCHEMBL2892834 0.81 ITGB1 (0.41) ITGB1ITGA4ITGB7CTSCTACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed