SCHEMBL1647997

SCHEMBL1647997

O=C(/C=C/c1ccc(O)cc1)CC(=O)/C=C/c1cc(OCc2ccccc2)ccc1-c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 14/20 1.00
GSK3B P49841 4/20 0.66
ABCG2 Q9UNQ0 1/20 0.57
SLC5A1 P13866 1/20 0.52
SLC5A2 P31639 1/20 0.52
APP P05067 2/20 0.50
MAPT P10636 1/20 0.50
CYP1A1 P04798 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP19A1 P11511 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1648000 1.00 BACE1 (1.00) BACE1GSK3BABCG2SLC5A1SLC5A2
SCHEMBL1646670 0.86 BACE1 (0.77) BACE1GSK3BABCG2SLC5A1SLC5A2
SCHEMBL1646956 0.86 BACE1 (1.00) BACE1GSK3BABCG2SLC5A1SLC5A2
SCHEMBL1646677 0.86 BACE1 (0.77) BACE1GSK3BABCG2SLC5A1SLC5A2
SCHEMBL1646957 0.86 BACE1 (1.00) BACE1GSK3BABCG2SLC5A1SLC5A2
SCHEMBL1648281 0.85 BACE1 (1.00) BACE1
SCHEMBL1648285 0.85 BACE1 (1.00) BACE1
SCHEMBL1646337 0.85 BACE1 (0.73) BACE1GSK3BAPPMAPT
SCHEMBL1646332 0.85 BACE1 (0.73) BACE1GSK3BAPPMAPT
SCHEMBL1645624 0.83 APP (0.73) BACE1GSK3BAPPMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8962674-B2 Curcumin derivative TOKYO INSTITUTE OF TECHNOLOGY (JP) 2015-02-24 US disclosed
US-8552220-B2 Therapeutic agent for Alzheimer's disease TOKYO INSTITUTE OF TECHNOLOGY (JP) 2013-10-08 US disclosed
EP-2305629-A1 THERAPEUTIC AGENT FOR ALZHEIMER'S DISEASE Tokyo Institute of Technology (JP) 2011-04-06 EP disclosed
US-20100048901-A1 NOVEL CURCUMIN DERIVATIVE TOKYO INSTITUTE OF TECHNOLOGY (JP) 2010-02-25 US disclosed
EP-2123637-A1 NOVEL CURCUMIN DERIVATIVE Tokyo Institute of Technology (JP) 2009-11-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048901-A1 NOVEL CURCUMIN DERIVATIVE BACE1, APP, BACE2 BACE1 1/4885GSK3B 851/4885ABCG2 3722/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.