SCHEMBL16480412

SCHEMBL16480412

CNC(=O)c1cccc(N2C(=O)CCC2C)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
RAB9A P51151 4/20 0.44
NPC1 O15118 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
L3MBTL3 Q96JM7 1/20 0.43
KDM4E B2RXH2 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
ABL1 P00519 2/20 0.41
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.41
P2RX3 P56373 1/20 0.41
P2RX2 Q9UBL9 1/20 0.41
MAPT P10636 1/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28804472 0.85 PARP1 (0.49) MEN1KMT2ARAB9AALDH1A1L3MBTL1
SCHEMBL16542508 0.85 ALDH1A1 (0.54) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL2570464 0.85 MEN1 (0.55) MEN1KMT2AHDAC8HDAC6RAB9A
SCHEMBL2570466 0.85 MEN1 (0.55) MEN1KMT2AHDAC8HDAC6RAB9A
SCHEMBL16480486 0.84 GAA (0.53) KMT2ARAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL9893047 0.84 MEN1 (0.54) MEN1KMT2AHDAC8HDAC6RAB9A
SCHEMBL9891741 0.84 MEN1 (0.54) MEN1KMT2AHDAC8HDAC6RAB9A
SCHEMBL16480487 0.83 HDAC2 (0.46) MEN1KMT2AHDAC8HDAC6RAB9A
SCHEMBL16480488 0.82 PMM2 (0.45) MEN1KMT2ANPC1SMN1; SMN2ALDH1A1
SCHEMBL16480394 0.76 KMT2A (0.48) MEN1KMT2AALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8629157-B2 Pyrrolidine compounds which modulate the CB2 receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-14 US disclosed