SCHEMBL16480490

SCHEMBL16480490

COc1ccc(N2C(=O)CCC2C)nc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.40
TNF P01375 1/20 0.39
ALDH1A1 P00352 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LCAT P04180 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
ABL1 P00519 2/20 0.37
IDH1 O75874 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GRM5 P41594 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9891785 0.83 HRH3 (0.44) HRH3ALDH1A1L3MBTL1KDM4EMAPT
SCHEMBL9108258 0.82 IDH1 (0.43) HRH3ALDH1A1L3MBTL1KDM4EPOLB
SCHEMBL9108249 0.82 IDH1 (0.43) HRH3ALDH1A1L3MBTL1KDM4EPOLB
SCHEMBL16480457 0.82 NPC1 (0.45) HRH3ALDH1A1NPSR1ABL1
SCHEMBL9893027 0.81 GRM5 (0.42) HRH3ABL1GRM5
SCHEMBL13285315 0.81 GRIN2D (0.38) HRH3MAPTABL1GRM5
SCHEMBL9893029 0.81 GAA (0.44) ALDH1A1KDM4EMAPTNPSR1CYP1A2
SCHEMBL9892984 0.78 POLB (0.54) ALDH1A1L3MBTL1POLBCYP1A2CYP3A4
SCHEMBL9892997 0.77 MAPT (0.51) HRH3ALDH1A1L3MBTL1KDM4EMAPT
SCHEMBL9893014 0.77 CNR1 (0.50) ALDH1A1L3MBTL1KDM4EGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2384320-B1 PYRROLIDINE COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INT (DE) 2015-03-04 EP disclosed
US-8629157-B2 Pyrrolidine compounds which modulate the CB2 receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-14 US disclosed