SCHEMBL1648331

SCHEMBL1648331

Cn1ccc(-c2ccc(OCc3ccc(F)cc3)c(C(=O)Nc3ccnnc3)c2)n1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 20/20 0.59
SRPK3 Q9UPE1 1/20 0.51
CYP3A4 P08684 2/20 0.51
SLCO1B1 Q9Y6L6 2/20 0.51
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1648615 0.86 LRRK2 (0.79) LRRK2CYP3A4SLCO1B1KCNH2
SCHEMBL1647109 0.84 LRRK2 (0.65) LRRK2SRPK3CYP3A4SLCO1B1
SCHEMBL1647847 0.84 LRRK2 (0.79) LRRK2SRPK3CYP3A4SLCO1B1
SCHEMBL1647748 0.81 LRRK2 (0.81) LRRK2SRPK3CYP3A4SLCO1B1
SCHEMBL10322017 0.79 LRRK2 (0.60) LRRK2SRPK3CYP3A4SLCO1B1
SCHEMBL10820439 0.79 LRRK2 (0.83) LRRK2SRPK3CYP3A4SLCO1B1
SCHEMBL6917702 0.77 LRRK2 (0.67) LRRK2CYP3A4SLCO1B1KCNH2
SCHEMBL1646947 0.77 LRRK2 (0.61) LRRK2CYP3A4SLCO1B1KCNH2
SCHEMBL6918692 0.76 LRRK2 (0.80) LRRK2CYP3A4SLCO1B1KCNH2
SCHEMBL6917773 0.76 LRRK2 (0.65) LRRK2CYP3A4SLCO1B1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483254-A1 NOVEL COMPOUNDS Glaxo Group Limited (GB) 2012-08-08 EP disclosed
WO-2011038572-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-04-07 WO disclosed