SCHEMBL1648795

SCHEMBL1648795

COc1cccc(CNC(=O)c2cnn3cc(-c4cn[nH]c4)ccc23)c1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 16/20 0.68
ROCK1 Q13464 10/20 0.68
PRKACA P17612 5/20 0.64
PRKACG P22612 5/20 0.64
PRKACB P22694 5/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23384715 0.88 ROCK2 (0.51) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1649829 0.87 ROCK2 (0.65) ROCK2ROCK1PRKACA
SCHEMBL1647289 0.81 ROCK2 (0.79) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL23384934 0.81 PRKACA (0.66) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL15968147 0.81 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL18685145 0.81 ROCK2 (0.81) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL3812995 0.80 ROCK2 (0.76) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL18685098 0.80 ROCK2 (0.80) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL17439838 0.80 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL17439778 0.80 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed