Bicarbonate

Bicarbonate

SCHEMBL16493752

CO[C@H]1CC[C@H](NC(=O)c2ccc(-c3ccccc3Cl)c(-c3ccc(Cl)c(OCCCN(C)C)c3)n2)CC1.Cl.O=C(O)O

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.42
CNR1 P21554 4/20 0.39
PAICS P22234 1/20 0.37
BRD4 O60885 2/20 0.37
UTS2R Q9UKP6 1/20 0.37
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR6 P50406 1/20 0.36
ATM Q13315 1/20 0.36
SLC6A9 P48067 2/20 0.36
CNR2 P34972 5/20 0.36
GABRA1 P14867 1/20 0.35
FAAH O00519 2/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL16493685 1.00 HTR7 (0.42) HTR7CNR1PAICSBRD4UTS2R
Bicarbonate SCHEMBL16493677 0.93 HTR7 (0.43) HTR7CNR1PAICSBRD4UTS2R
Bicarbonate SCHEMBL16493849 0.92 CNR1 (0.48) HTR7CNR1ATMCNR2FAAH
Hydrochloric Acid SCHEMBL544475 0.87 PAICS (0.36) HTR7PAICSATMSLC6A9KDM4E
Hydrochloric Acid SCHEMBL544474 0.87 PAICS (0.36) HTR7PAICSATMSLC6A9KDM4E
Hydrochloric Acid SCHEMBL4046584 0.87 PAICS (0.36) HTR7PAICSATMSLC6A9KDM4E
Hydrochloric Acid SCHEMBL544476 0.87 PAICS (0.36) HTR7PAICSATMSLC6A9KDM4E
Bicarbonate SCHEMBL16493748 0.87 HTR7 (0.42) HTR7CNR1PAICSBRD4UTS2R
Bicarbonate SCHEMBL16493561 0.87 ATM (0.42) HTR7CNR1PAICSUTS2RHTR1A
Bicarbonate SCHEMBL16493556 0.87 HTR7 (0.42) HTR7CNR1PAICSBRD4UTS2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2059508-B1 5,6-BISARYL-2-PYRIDINE-CARBOXAMIDE DERIVATIVES, PREPARATION AND APPLICATION THEREOF IN THERAPEUTICS AS UROTENSIN II RECEPTOR ANTAGONISTS SANOFI SA (FR) 2012-04-11 EP claimed