SCHEMBL164941

SCHEMBL164941

Fc1ccc(Br)cc1.[MgH2]

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7026005 0.96
SCHEMBL29525203 0.96
SCHEMBL1622 0.96
Fluoride SCHEMBL27504442 0.93 CYP2A6 (0.57)
SCHEMBL28116949 0.93
Fluoride SCHEMBL25376004 0.93 CYP2A6 (0.57)
SCHEMBL27470752 0.93
SCHEMBL4600807 0.93
Water SCHEMBL28292373 0.93
SCHEMBL8863391 0.91 MAPK1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1352 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120058632-A Method for synthesizing aprepitant intermediate through hydrogenation 苏州乔贝迪医药科技有限公司 2025-05-30 CN claimed
CN-119798292-A Polycyclic fusion molecule containing oxygen, boron and nitrogen coordination bonds and preparation method thereof 华侨大学 2025-04-11 CN claimed
CN-119285931-A Preparation method of polyarylether phosphine oxide intrinsic type room temperature phosphorescent material 重庆理工大学 2025-01-10 CN claimed
CN-118908996-A A composition containing C (sp2) P bond or C (sp)3) Process for preparing organic phosphine compound of-P bond 烟台大学 2024-11-08 CN claimed
CN-114874080-B Preparation method of 4,4' -difluorobenzophenone 绍兴久孚新材料科技有限公司 2024-08-02 CN claimed
CN-114380870-B Preparation method and application of homogeneous cobalt chloride/tetramethyl ethylenediamine complex solution 山东东岳高分子材料有限公司 2024-06-28 CN claimed
CN-114409602-B Method for synthesizing alpha-keto acid by using oxalyl chloride and Grignard reagent as raw materials 武汉大学 2024-01-30 CN claimed
WO-2023124996-A1 SULFUR-CONTAINING CHIRAL BRIDGED METALLOECENE COMPOUND, PREPARATION THEREOF, AND APPLICATION 中国石油天然气股份有限公司 2023-07-06 WO claimed
CN-113620869-B Preparation method of betrixaban 江西同和药业股份有限公司 2023-04-18 CN claimed
CN-112409212-B Preparation method of citalopram diol intermediate hydrobromide, citalopram diol intermediate hydrobromide and citalopram 四川新迪医药化工有限公司 2023-03-14 CN claimed
US-20030153774-A1 Process for the preparation of citalopram PHARMACHEM TECHNOLOGIES LIMITED, (GB) 2003-08-14 US claimed
US-20030130527-A1 Process for the preparation of 1-(3-dimethylaminopropyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-carbonitrile ORION CORPORATION FERMION (FI) 2003-07-10 US claimed
US-6579993-B2 Halogenating 5-cyanophthalide to a cyanobenzeneacyl halide derivative reacted with organometallic 4-fluorophenyl halides and 4-fluorophenylboranes to a biphenyl ketone reacted with an organometallic 3-dimethylaminopropyl halide ORION CORPORATION, FERMION (FI) 2003-06-17 US claimed
WO-2003040121-A1 METHODS FOR TREATING DEPRESSION AND OTHER CNS DISORDERS USING ENANTIOMERICALLY ENRICHED DESMETHYL- AND DIDESMETHYL-METABOLITES OF CITALOPRAM SEPRACOR, INC. (US) 2003-05-15 WO claimed
WO-2003029236-A1 PROCESS FOR THE PREPARATION OF CITALOPRAM PHARMACHEM TECHNOLOGIES LIMITED (GB) 2003-04-10 WO claimed
US-20020115872-A1 Process for the preparation of 1-(3-dimethylaminopropyl)-1-(4-Fluorophenyl)-1,3-dihydroisobenzofuran-5-carbonitrile ORION CORPORATION FERMION (FI) 2002-08-22 US claimed
WO-2002060886-A1 PROCESS FOR THE PREPARATION OF 1-(3-DIMETHYLAMINOPROPYL)-1-(4-FLUOROPHENYL)-1,3-DIHYDROISOBENZOFURAN-5-CARBONITRILE ORION CORPORATION, FERMION (FI) 2002-08-08 WO claimed
CN-1331685-A Process for the preparation of citalopram LUNDBECK & CO AS H (DK) 2002-01-16 CN claimed
EP-1064286-A1 SYNTHESIS OF ARYL BORONIC ACIDS BOULDER SCIENTIFIC COMPANY (US) 2001-01-03 EP claimed
WO-1999064428-A1 SYNTHESIS OF ARYL BORONIC ACIDS BOULDER SCIENTIFIC COMPANY (US) 1999-12-16 WO claimed