SCHEMBL16494261

SCHEMBL16494261

Nc1ccc(Cl)nc1NC1CCN(C(=O)O)CC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 10/20 0.39
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
SLC6A12 P48065 1/20 0.37
BTK Q06187 3/20 0.36
EGFR P00533 1/20 0.36
CNR1 P21554 3/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1694560 0.82 ALDH1A1 (0.55) BTKCNR1MEN1MAPTHTT
SCHEMBL20337764 0.81 ACP1 (0.38) KDM4EMAPTKMT2A
SCHEMBL29526189 0.81 ACP1 (0.38) KDM4EMAPTKMT2A
SCHEMBL19691685 0.81 EGFR (0.40) PAK1NOS1NOS2BTKEGFR
SCHEMBL1783130 0.81 KMT2A (0.43) PAK1NOS1NOS2BTKEGFR
SCHEMBL1693347 0.80 MAPT (0.52) MEN1MAPTHTTKMT2A
SCHEMBL1693350 0.80 MAPT (0.52) MEN1MAPTHTTKMT2A
SCHEMBL12936052 0.78 KDM4E (0.43) KDM4EMEN1MAPTKMT2A
SCHEMBL27907279 0.78 SSTR4 (0.37) PAK1NOS1NOS2SLC6A12BTK
SCHEMBL14768725 0.77 KMT2A (0.45) KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2397482-A1 Heteroaryl imidazolone derivatives as jak inhibitors Almirall, S.A. (ES) 2011-12-21 EP disclosed