SCHEMBL16498403

SCHEMBL16498403

C[C@@H](NC(=O)O)C(=O)Nc1ccc(-c2ccncc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.58
PSEN1 P49768 4/20 0.51
PSEN2 P49810 4/20 0.51
APH1B Q8WW43 4/20 0.51
NCSTN Q92542 4/20 0.51
APH1A Q96BI3 4/20 0.51
PSENEN Q9NZ42 4/20 0.51
TAAR1 Q96RJ0 1/20 0.49
ROCK2 O75116 7/20 0.48
CYP3A4 P08684 1/20 0.48
CYP3A5 P20815 1/20 0.48
ROCK1 Q13464 6/20 0.48
LMNA P02545 1/20 0.46
RPS6KA5 O75582 1/20 0.46
MAP4K4 O95819 1/20 0.46
CDK1 P06493 1/20 0.46
CSF1R P07333 1/20 0.46
PRKACA P17612 1/20 0.46
FLT1 P17948 1/20 0.46
RPS6KB1 P23443 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16512502 0.88 AAK1 (0.61) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL4535633 0.82 AAK1 (0.56) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL10259810 0.82 AAK1 (0.56) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL27723715 0.82 AAK1 (0.56) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL16370847 0.82 AAK1 (0.66) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL16371179 0.82 AAK1 (0.59) AAK1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL4520449 0.81 AAK1 (0.54) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL16512501 0.81 CYP17A1 (0.58) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL11187399 0.81 AAK1 (0.64) AAK1PSEN1PSEN2APH1BNCSTN
SCHEMBL4516268 0.78 ROCK2 (0.57) AAK1TAAR1ROCK2ROCK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011153588-A1 VIRAL POLYMERASE INHIBITORS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2011-12-15 WO disclosed