SCHEMBL16500166

SCHEMBL16500166

[c]1nc2cc(-c3ccc4c(c3)nc(-c3ccccc3)n4Nc3ccccc3)ccc2[nH]1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NLRP3 Q96P20 1/20 0.33
NAMPT P43490 1/20 0.32
PDE10A Q9Y233 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALK Q9UM73 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409270 0.75 DYRK3 (0.43) KDM4ENPC1GAAALK
SCHEMBL27947333 0.64 FGFR1 (0.43) KDM4ENPC1GAA
SCHEMBL16500231 0.64 NPC1 (0.43) HDAC1HDAC8HDAC6KDM4ENPC1
SCHEMBL699438 0.63 MAP4K4 (0.36) KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20412071 0.63 PDE3B (0.46) ALK
SCHEMBL27847161 0.62 PDPK1 (0.44)
SCHEMBL1104828 0.62 HDAC1 (0.64) HDAC1HDAC8HDAC6NLRP3NAMPT
SCHEMBL3103036 0.61 NQO2 (0.43) KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL28013699 0.61 KMT2A (0.58) GAARAB9ASMN1; SMN2
SCHEMBL29062356 0.60 KMT2A (0.41) KDM4ECYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373631-B1 ANTIBACTERIAL COMPOUNDS SUMMIT CORP PLC (GB) 2015-02-25 EP claimed