SCHEMBL16503564

SCHEMBL16503564

Bc1ccc(S(=O)(=O)N2CCC[C@@H]2CO)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.57
BRD2 P25440 1/20 0.57
PSEN1 P49768 2/20 0.50
PSEN2 P49810 2/20 0.50
APH1B Q8WW43 2/20 0.50
NCSTN Q92542 2/20 0.50
APH1A Q96BI3 2/20 0.50
PSENEN Q9NZ42 2/20 0.50
PLAU P00749 1/20 0.48
LOX P28300 1/20 0.48
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
NAMPT P43490 2/20 0.47
HTR7 P34969 1/20 0.44
TRPA1 O75762 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4610414 0.87 BRD4 (0.58) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL6302770 0.85 BRD4 (0.57) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL5885963 0.85 BRD4 (0.57) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL5885959 0.85 BRD4 (0.57) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL1684457 0.85 BRD4 (0.57) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL1684459 0.85 BRD4 (0.57) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL15256572 0.85 BRD4 (0.57) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL19563388 0.85 BRD4 (0.57) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL28243010 0.85 TRPA1 (0.61) BRD4BRD2PSEN1PSEN2APH1B
SCHEMBL17600734 0.85 BRD4 (0.56) BRD4BRD2PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2395002-A1 Pharmaceutical composition containing a heterocyclic modulator of ATP-binding cassette transporters. Vertex Pharmaceuticals Incorporated (US) 2011-12-14 EP disclosed