Mertiatide

Mertiatide

SCHEMBL1650428

O=C(O)CNC(=O)CNC(=O)CNC(=O)CS.O=[99Tc]

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
MAPT P10636 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
LMNA P02545 1/20 0.39
PTGS2 P35354 1/20 0.39
MME P08473 7/20 0.37
EGLN1 Q9GZT9 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
FAAH O00519 5/20 0.34
ACE P12821 3/20 0.33
CPA1 P15085 1/20 0.33
ACE2 Q9BYF1 1/20 0.33
PTPN1 P18031 1/20 0.33
PTGS1 P23219 1/20 0.33
GSTK1 Q9Y2Q3 1/20 0.33
MEN1 O00255 2/20 0.33
HPGD P15428 2/20 0.33
BLM P54132 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mertiatide SCHEMBL136462 0.95 ALDH1A1 (0.41) ALDH1A1MAPTTDP1LMNAPTGS2
SCHEMBL1493216 0.95 ALDH1A1 (0.41) ALDH1A1MAPTTDP1LMNAPTGS2
SCHEMBL14417106 0.95 ALDH1A1 (0.41) ALDH1A1MAPTTDP1LMNAPTGS2
Mertiatide SCHEMBL23522195 0.93 ALDH1A1 (0.40) ALDH1A1MAPTTDP1LMNAPTGS2
SCHEMBL2796838 0.93 ALDH1A1 (0.40) ALDH1A1MAPTTDP1LMNAPTGS2
SCHEMBL75812 0.91
SCHEMBL12762758 0.84 ALDH1A1 (0.34) ALDH1A1MAPTTDP1LMNAPTGS2
Glycine SCHEMBL4653213 0.82 GLRA1 (0.46) ALDH1A1MAPTTDP1LMNAPTGS2
Glycine SCHEMBL4264488 0.82 GLRA1 (0.46) ALDH1A1MAPTTDP1LMNAPTGS2
SCHEMBL610938 0.80 ALDH1A1 (0.38) ALDH1A1MAPTTDP1LMNAPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
US-7790905-B2 Pharmaceutical propylene glycol solvate compositions MCNEIL-PPC, INC. (US) 2010-09-07 US disclosed