SCHEMBL16517536

SCHEMBL16517536

NC(=O)c1c2cccnc2nn1-c1cc(Br)cc(N2CCOCC2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
PIK3R2 O00459 1/20 0.37
PIK3CA P42336 5/20 0.37
MTOR P42345 4/20 0.37
PIK3CD O00329 3/20 0.37
PIK3CG P48736 2/20 0.37
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LMNA P02545 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
ABCB1 P08183 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
PIK3R1 P27986 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16516729 0.91 KMO (0.39) PIK3CAMTORPIK3CDPIK3CGSMN1; SMN2
SCHEMBL16517270 0.87 MRGPRX4 (0.39) PIK3CAMTORPIK3CDPIK3CGGAA
SCHEMBL16532453 0.82 MAP3K14 (0.46) AURKARPS6KB1MAPK9MAPK10LRRK2
SCHEMBL16516862 0.79 PDE4A (0.51) AURKARPS6KB1GAAKDM4EALDH1A1
SCHEMBL16517092 0.79 MAP3K14 (0.40) GAASMN1; SMN2KDM4EALDH1A1PDE4A
SCHEMBL16517022 0.77 MAOB (0.38) AURKARPS6KB1KDM4EPDE4ATYK2
SCHEMBL16532395 0.73 MAPT (0.45) GAASMN1; SMN2MAPK10ABCB1KDM4E
SCHEMBL16517380 0.69 RPA1 (0.40) AURKASMN1; SMN2NPSR1ALDH1A1HTT
SCHEMBL16516797 0.69 PDE4A (0.44) AURKASMN1; SMN2KDM4EALDH1A1PDE4A
SCHEMBL30099106 0.68 KMO (0.48) PIK3CAPIK3CDPIK3CGSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3036230-A1 ALKYNYL ALCOHOLS AND METHODS OF USE F. Hoffmann-La Roche AG (CH) 2016-06-29 EP disclosed
WO-2015025025-A1 ALKYNYL ALCOHOLS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2015-02-26 WO disclosed