SCHEMBL16588387

SCHEMBL16588387

O=C1NCCN1CCCNI

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.42
ALDH1A1 P00352 4/20 0.42
RAB9A P51151 1/20 0.42
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 3/20 0.39
MEN1 O00255 3/20 0.37
MAPT P10636 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RET P07949 1/20 0.35
KDR P35968 1/20 0.35
CREBBP Q92793 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16588388 0.89 KMT2A (0.48) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL13843636 0.82 ALDH1A1 (0.47) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL7261352 0.82 ALDH1A1 (0.47) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL6287263 0.81 KMT2A (0.46) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL1446116 0.80 ALDH1A1 (0.43) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL14426104 0.80 KMT2A (0.41) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL2118226 0.80 ALDH1A1 (0.46) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL11173610 0.80 ALDH1A1 (0.46) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL6285538 0.79 KMT2A (0.43) KMT2AALDH1A1RAB9AKDM4ELMNA
SCHEMBL4465738 0.79 KMT2A (0.40) KMT2AALDH1A1RAB9AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2625169-B1 QUINAZOLINE COMPOUNDS AS SODIUM CHANNEL BLOCKERS PURDUE PHARMA LP (US) 2015-03-25 EP disclosed