SCHEMBL16600111

SCHEMBL16600111

NC(=O)c1c(F)c(F)c(-c2ccccc2)c(N2CCNCC2)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.41
HTR2C P28335 2/20 0.41
HTR6 P50406 3/20 0.40
PARP1 P09874 1/20 0.39
ALDH1A1 P00352 2/20 0.39
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HTR7 P34969 3/20 0.38
HTR1A P08908 2/20 0.38
HTR5A P47898 1/20 0.38
OPRD1 P41143 1/20 0.38
SIGMAR1 Q99720 2/20 0.37
LMNA P02545 1/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
ADRB1 P08588 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16599761 0.86 HTR2A (0.39) HTR2AHTR2CHTR6PARP1ALDH1A1
SCHEMBL9042452 0.72 HTR6 (0.40) HTR2AHTR2CHTR6ALDH1A1USP2
SCHEMBL20527676 0.72 HTR6 (0.40) HTR2AHTR6ALDH1A1USP2TSHR
SCHEMBL9042443 0.72 HTR6 (0.40) HTR2AHTR2CHTR6ALDH1A1USP2
SCHEMBL14746666 0.71 PTPN11 (0.57) HTR2AHTR6ALDH1A1TSHRHSD17B10
SCHEMBL6651301 0.70 HTR6 (0.44) HTR2AHTR2CHTR6ALDH1A1USP2
SCHEMBL14746663 0.70 HRH4 (0.40) HTR2CHTR6PARP1ALDH1A1USP2
SCHEMBL4918486 0.70 HTR6 (0.50) HTR2AHTR2CHTR6ALDH1A1TSHR
SCHEMBL379430 0.69 HTR6 (0.51) HTR2AHTR6PARP1ALDH1A1TSHR
SCHEMBL6746969 0.69 ACVR1 (0.41) HTR2AHTR6ALDH1A1USP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015048306-A1 NOVEL AGENTS TARGETING CYP51 THE SCRIPPS RESEARCH INSTITUTE (US) 2015-04-02 WO disclosed