SCHEMBL1660015

SCHEMBL1660015

CCC(C(=O)O)n1nc(-c2cccc(C3(NC(=O)OC(C)(C)C)COC3)c2)cc1Oc1ccc(C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.36
P2RY14 Q15391 2/20 0.34
SCN9A Q15858 4/20 0.33
PIK3CD O00329 1/20 0.32
PIK3C2B O00750 1/20 0.32
MAP2K4 P45985 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
RXRA P19793 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
SUCNR1 Q9BXA5 2/20 0.31
BRD9 Q9H8M2 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
PTGER4 P35408 1/20 0.31
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1660744 0.88 PDE2A (0.38) PDE2AP2RY14SCN9APIK3CDPIK3C2B
SCHEMBL14727913 0.86 TRPM2 (0.37) PDE2AP2RY14SCN9APIK3CDPIK3C2B
SCHEMBL6903422 0.85 PDE2A (0.34) PDE2AP2RY14SCN9APIK3CDPIK3C2B
SCHEMBL6903551 0.84 PDE2A (0.36) PDE2AP2RY14SCN9APIK3CDPIK3C2B
SCHEMBL6904357 0.81 SRPK1 (0.36) PDE2ASCN9APIK3CD
SCHEMBL6903557 0.79 PDE2A (0.40) PDE2AP2RY14SCN9AMAP2K4SCN10A
SCHEMBL14717866 0.79 PDE2A (0.39) PDE2AP2RY14SCN9APIK3CDSCN10A
SCHEMBL14718861 0.77 PDE2A (0.37) PDE2ASCN9ASCN10A
SCHEMBL6902906 0.76 TRPM2 (0.37) PDE2ASCN9APIK3CDSCN10A
SCHEMBL11962993 0.76 PDE2A (0.40) PDE2AP2RY14SCN9ASCN10APTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046774-A1 DIARYL ETHER DERIVATIVES AS NOTCH SPARING GAMMA SECRETASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-04-21 WO disclosed