SCHEMBL16600415

SCHEMBL16600415

O=C(O)c1cccc(Sc2c(C3CC3)n(CC(=O)N3CCc4ccccc43)c3c(F)c(Cl)ccc23)c1F.[NaH]

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 17/20 0.63
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
RAB9A P51151 1/20 0.43
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16614212 0.99 ENPP2 (0.64) ENPP2NPC1ALDH1A1RAB9ANPSR1
SCHEMBL16600414 0.92 ENPP2 (0.61) ENPP2NPC1ALDH1A1RAB9ANPSR1
SCHEMBL16600530 0.89 ENPP2 (0.58) ENPP2ALDH1A1
SCHEMBL16600463 0.88 ENPP2 (0.61) ENPP2NPC1ALDH1A1RAB9A
SCHEMBL17943014 0.87 ENPP2 (0.61) ENPP2NPC1ALDH1A1RAB9A
SCHEMBL16600464 0.85 ENPP2 (0.81) ENPP2
SCHEMBL16614230 0.83 ENPP2 (0.77) ENPP2
SCHEMBL16600461 0.81 ENPP2 (0.54) ENPP2ALDH1A1
SCHEMBL17943189 0.80 ENPP2 (0.85) ENPP2
SCHEMBL16600595 0.79 ENPP2 (0.65) ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3049405-A1 AUTOTAXIN INHIBITOR COMPOUNDS Pharmakea Inc. (US) 2016-08-03 EP disclosed
WO-2015048301-A1 AUTOTAXIN INHIBITOR COMPOUNDS PHARMAKEA, INC. (US) 2015-04-02 WO disclosed