SCHEMBL16601597

SCHEMBL16601597

Cc1ccc2c(c1)oc(=O)n2CC(N)=O

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.64
MIF P14174 3/20 0.58
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPK1 P28482 1/20 0.47
TP53 P04637 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PKM P14618 1/20 0.45
CD74 P04233 1/20 0.45
PTGS2 P35354 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16250472 0.88 HPGD (0.64) HPGDMIFL3MBTL1RAB9ASMN1; SMN2
SCHEMBL5302441 0.87 MIF (0.63) MIFCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL14564389 0.83 MIF (0.56) MIFCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4411794 0.82 HPGD (0.64) HPGDSMN1; SMN2MAPK1TP53MEN1
SCHEMBL4413144 0.82 HPGD (0.64) HPGDMIFSMN1; SMN2MAPK1TP53
SCHEMBL4414360 0.82 HPGD (0.64) HPGDCYP3A4TP53MEN1KMT2A
SCHEMBL13340920 0.82 HPGD (0.59) HPGDSMN1; SMN2MAPK1TP53MEN1
SCHEMBL4413088 0.82 HPGD (0.59) HPGDSMN1; SMN2TP53KMT2A
SCHEMBL13367743 0.80 MIF (0.66) MIFL3MBTL1RAB9ASMN1; SMN2MEN1
SCHEMBL4414345 0.78 HPGD (1.00) HPGDMIFSMN1; SMN2MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8993585-B2 Cyclic amine substituted pyrimidinediamines as PKC inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-03-31 US disclosed